Oral Presentation Australian and New Zealand Obesity Society Annual Scientific Conference 2026

GLP-1 engages a dorsal raphe-preoptic 5-HT2C circuit to suppress drinking (144963)

Tiemin Liu 1 2 3
  1. State Key Laboratory of Genetics and Development of Complex Phenotypes, School of Life Sciences, Fudan University, Shanghai, CHINA
  2. Institutes of Biomedical Sciences, School of Life Sciences, Inner Mongolia University, Hohhot, Inner Mongolia Autonomous Region, CHINA
  3. Department of Endocrinology and Metabolism, Zhongshan Hospital, Human Phenome Institute,, Fudan University, Shanghai, CHINA

Abstract

Glucagon-like peptide-1 (GLP-1) receptor agonists are widely used to treat obesity and metabolic disease by suppressing food intake, yet their effects on fluid homeostasis remain poorly understood. Here we show that the GLP-1 analogue semaglutide robustly suppresses water intake in mice independently of its anorexigenic action, revealing an unexpected role for GLP-1 signaling in the control of drinking behavior. Semaglutide activates serotonergic neurons in the dorsal raphe nucleus (DRN), resulting in serotonin-mediated inhibition of 5-HT2C receptor–expressing neurons in the medial preoptic area (MPA). These MPA 5-HT2C neurons are activated immediately prior to drinking and encode an aversive motivational state; their chemogenetic or optogenetic activation induces excessive water intake, whereas their inhibition suppresses drinking. Conversely, genetic deletion of Htr2c in the MPA disinhibits this population, elevates basal water consumption, and abolishes semaglutide-induced suppression of drinking without affecting appetite regulation. Together, these findings identify a serotonin-modulated DRNàMPA circuit that selectively governs thirst and demonstrate that GLP-1 mediated suppression of drinking is mechanistically distinct from feeding suppression. This work uncovers a previously unrecognized dimension of GLP-1 signaling with implications for fluid balance regulation during anti-obesity therapy.